| 1 |
Synthesis and antimicrobial activities of novel quinoline derivatives carrying 1,2,4-triazole moiety
Sumesh Eswaran, Airody Vasudeva Adhikari, N. Suchetha Shetty · European Journal of Medicinal Chemistry
|
4 Jul 2009 |
302 |
| 2 |
New quinoline derivatives: Synthesis and investigation of antibacterial and antituberculosis properties
Sumesh Eswaran, Airody Vasudeva Adhikari, Imran Hussain Chowdhury et al. · European Journal of Medicinal Chemistry
|
29 Apr 2010 |
222 |
| 3 |
Liquid-Phase Peptide Synthesis (LPPS): A Third Wave for the Preparation of Peptides
Anamika Sharma, Ashish Kumar, Beatriz Garcia de la Torre et al. · Chemical Reviews
ReviewOpen access |
11 Jul 2022 |
161 |
| 4 |
Design, synthesis and antimicrobial activities of some new quinoline derivatives carrying 1,2,3-triazole moiety
K.D. Thomas, Airody Vasudeva Adhikari, N. Suchetha Shetty · European Journal of Medicinal Chemistry
|
21 May 2010 |
145 |
| 5 |
Biomimetic Iron‐Catalyzed Asymmetric Epoxidation of Aromatic Alkenes by Using Hydrogen Peroxide
Feyissa Gadissa Gelalcha, Gopinathan Nair Anilkumar, Man Kin Tse et al. · Chemistry - A European Journal
|
20 Jun 2008 |
136 |
| 6 |
Design, synthesis and docking studies of new quinoline-3-carbohydrazide derivatives as antitubercular agents
K.D. Thomas, Airody Vasudeva Adhikari, Sandeep B. Telkar et al. · European Journal of Medicinal Chemistry
|
29 Jul 2011 |
116 |
| 7 |
New quinolin-4-yl-1,2,3-triazoles carrying amides, sulphonamides and amidopiperazines as potential antitubercular agents
K.D. Thomas, Airody Vasudeva Adhikari, Imran Hussain Chowdhury et al. · European Journal of Medicinal Chemistry
|
15 Apr 2011 |
101 |
| 8 |
New 1,3-oxazolo[4,5-c]quinoline derivatives: Synthesis and evaluation of antibacterial and antituberculosis properties
Sumesh Eswaran, Airody Vasudeva Adhikari, R. Ajay Kumar · European Journal of Medicinal Chemistry
|
28 Nov 2009 |
98 |
| 9 |
Design and synthesis of some new quinoline-3-carbohydrazone derivatives as potential antimycobacterial agents
Sumesh Eswaran, Airody Vasudeva Adhikari, Nishith Kumar Pal et al. · Bioorganic & Medicinal Chemistry Letters
|
17 Dec 2009 |
87 |
| 10 |
CRISPR/Cas-Based Modifications for Therapeutic Applications: A Review
Nagaraj Bharathkumar, Sunil Abraham, Prabhakar Meera et al. · Molecular Biotechnology
Open access |
6 Nov 2021 |
76 |
| 11 |
Drug Design and Disease Diagnosis: The Potential of Deep Learning Models in Biology
Sarojini Sreeraman, Kannan Mayuri, Raja Babu Singh Kushwah et al. · Current Bioinformatics
|
27 Feb 2023 |
70 |
| 12 |
Bibliometric analysis of artificial intelligence in healthcare research: Trends and future directions
Renganathan Senthil, Thirunavukarasou Anand, Chaitanya Sree Somala et al. · Future Healthcare Journal
Open access |
Sep 2024 |
69 |
| 13 |
Synthesis, antituberculosis studies and biological evaluation of new quinoline derivatives carrying 1,2,4-oxadiazole moiety
T. G. Shruthi, Sumesh Eswaran, Prasad Shivarudraiah et al. · Bioorganic & Medicinal Chemistry Letters
|
2 Nov 2018 |
69 |
| 14 |
Advancement of Targeted Protein Degradation Strategies As Therapeutics for Undruggable Disease Targets
Kannan Mayuri, Sarojini Sreeraman, Chaitanya Sree Somala et al. · Future Medicinal Chemistry
|
May 2023 |
62 |
| 15 |
An amide to thioamide substitution improves the permeability and bioavailability of macrocyclic peptides
Pritha Ghosh, Nishant Raj, Hitesh Verma et al. · Nature Communications
Open access |
28 Sep 2023 |
61 |
| 16 |
Antioxidant and nephroprotection activities of Combretum micranthum: A phytochemical, in-vitro and ex-vivo studies
Mabozou Kpemissi, Kwashie Eklu‐Gadegbeku, Veeresh Prabhakar Veerapur et al. · Heliyon
Open access |
Mar 2019 |
61 |
| 17 |
Nephroprotective activity of Combretum micranthum G. Don in cisplatin induced nephrotoxicity in rats: In-vitro, in-vivo and in-silico experiments
Mabozou Kpemissi, Kwashie Eklu‐Gadegbeku, Veeresh Prabhakar Veerapur et al. · Biomedicine & Pharmacotherapy
Open access |
28 May 2019 |
57 |
| 18 |
Pseudomonas aeruginosa virulence attenuation by inhibiting siderophore functions
Geum‐Jae Jeong, Fazlur-Rahman Nawaz Khan, Sohail Khan et al. · Applied Microbiology and Biotechnology
|
12 Jan 2023 |
55 |
| 19 |
Discovery of lesser known flavones as inhibitors of NF-κB signaling in MDA-MB-231 breast cancer cells—A SAR study
K. Amrutha, Pandurangan Nanjan, Sanu Korumadathil Shaji et al. · Bioorganic & Medicinal Chemistry Letters
|
13 Aug 2014 |
53 |
| 20 |
Design, synthesis and docking studies of quinoline-oxazolidinone hybrid molecules and their antitubercular properties
K.D. Thomas, Airody Vasudeva Adhikari, Imran Hussain Chowdhury et al. · European Journal of Medicinal Chemistry
|
Sep 2011 |
48 |
| 21 |
Design, Synthesis and Study of Antibacterial and Antitubercular Activity of Quinoline Hydrazone Hybrids
T. G. Shruthi, Sangeetha Subramanian, Sumesh Eswaran · Heterocyclic Communications
Open access |
2020 |
46 |
| 22 |
Zebrafish as an In Vivo High-Throughput Model for Genotoxicity
Sridhara Chakravarthy, Sathish Sadagopan, Ayyappan R. Nair et al. · Zebrafish
|
15 Jan 2014 |
45 |
| 23 |
Adaptation of Lactobacillus acidophilus to Thermal Stress Yields a Thermotolerant Variant Which Also Exhibits Improved Survival at pH 2
Sonia Kulkarni, Saiful F. Haq, Shalaka Samant et al. · Probiotics and Antimicrobial Proteins
|
29 Aug 2017 |
42 |
| 24 |
Impact of aqueous micellar media on biocatalytic transformations involving transaminase (ATA); applications to chemoenzymatic catalysis
Jade Dussart‐Gautheret, Tzu‐Yu Yu, Krithika Ganesh et al. · Green Chemistry
|
2022 |
38 |
| 25 |
Norspermidine and Novel Pd(II) and Pt(II) Polynuclear Complexes of Norspermidine as Potential Antineoplastic Agents Against Breast Cancer
Tânia Magalhães Silva, Sara Andersson, Sunil Kumar Sukumaran et al. · PLoS ONE
Open access |
13 Feb 2013 |
38 |
| 26 |
Fabrication of silver nanoparticles from marine macro algae Caulerpa sertularioides: Characterization, antioxidant and antimicrobial activity
Ravichandran Anjali, Subramanian Palanisamy, Manoharan Vinosha et al. · Process Biochemistry
|
27 Jul 2022 |
36 |
| 27 |
Syringaresinol as a novel androgen receptor antagonist against wild and mutant androgen receptors for the treatment of castration-resistant prostate cancer: molecular docking,in-vitroand molecular dynamics study
Divakar Selvaraj, Santhoshkumar Muthu, Satvik Kotha et al. · Journal of Biomolecular Structure and Dynamics
|
13 Jan 2020 |
35 |
| 28 |
Identifying Potent Fat Mass and Obesity-Associated Protein Inhibitors Using Deep Learning-Based Hybrid Procedures
Kannan Mayuri, Durairaj Varalakshmi, Mayakrishnan Tharaheswari et al. · BioMedInformatics
Open access |
Feb 2024 |
34 |
| 29 |
Effect of codon-optimized E. coli signal peptides on recombinant Bacillus stearothermophilus maltogenic amylase periplasmic localization, yield and activity
Shalaka Samant, Gunja Gupta, Subbulakshmi Karthikeyan et al. · Journal of Industrial Microbiology & Biotechnology
Open access |
19 Jul 2014 |
33 |
| 30 |
Whole cell screen based identification of spiropiperidines with potent antitubercular properties
Subramanyam Janardhan Tantry et al. · Bioorganic & Medicinal Chemistry Letters
Open access |
5 Jun 2015 |
33 |
| 31 |
ERK1/2 activated PHLPP1 induces skeletal muscle ER stress through the inhibition of a novel substrate AMPK
Soma Behera, Bandish B. Kapadia, Vasundhara Kain et al. · Biochimica et Biophysica Acta (BBA) - Molecular Basis of Disease
Open access |
27 Feb 2018 |
29 |
| 32 |
In situ Fmoc removal – a sustainable solid-phase peptide synthesis approach
Ashish Kumar, Anamika Sharma, Beatriz Garcia de la Torre et al. · Green Chemistry
Open access |
2022 |
27 |
| 33 |
New Hydroxamic Acid Derivatives of Fluoroquinolones: Synthesis and Evaluation of Antibacterial and Anticancer Properties
Gavara Govinda Rajulu, Halehatty S. Bhojya Naik, Abhilash Viswanadhan et al. · Chemical and Pharmaceutical Bulletin
Open access |
22 Nov 2013 |
27 |
| 34 |
Discovery of FNDR-20123, a histone deacetylase inhibitor for the treatment of Plasmodium falciparum malaria
Vijay Kumar Potluri, Radha Krishan Shandil, R. Gavara et al. · Malaria Journal
Open access |
12 Oct 2020 |
26 |
| 35 |
A multi-targeting pre-clinical candidate against drug-resistant tuberculosis
Parvinder Kaur, Vijay Kumar Potluri, Vijay Kamal Ahuja et al. · Tuberculosis
Open access |
18 Jun 2021 |
25 |
| 36 |
Kaposi's Sarcoma-Associated Herpesvirus-Positive Primary Effusion Lymphoma Tumor Formation in NOD/SCID Mice Is Inhibited by Neomycin and Neamine Blocking Angiogenin's Nuclear Translocation
Virginie Bottero, Sathish Sadagopan, Karen E. Johnson et al. · Journal of Virology
Open access |
29 Aug 2013 |
25 |
| 37 |
Safety assessment of Cissus quadrangularis extract (CQR-300): Subchronic toxicity and mutagenicity studies
Shil C. Kothari, Prasad Shivarudraiah, Suresh Babu Venkataramaiah et al. · Food and Chemical Toxicology
|
29 Sep 2011 |
25 |
| 38 |
Antibacterial efficacy of lytic phages against multidrug-resistant Pseudomonas aeruginosa infections in bacteraemia mice models
Shri Natrajan Arumugam, Prasanth Manohar, Sunilkumar Sukumaran et al. · BMC Microbiology
Open access |
Aug 2022 |
22 |
| 39 |
A strategy to identify a ketoreductase that preferentially synthesizes pharmaceutically relevant (S)-alcohols using whole-cell biotransformation
Saiful F. Haq, Anirudh P. Shanbhag, Subbulakshmi Karthikeyan et al. · Microbial Cell Factories
Open access |
Dec 2018 |
22 |
| 40 |
Design, synthesis and anti-cancer evaluation of a novel series of pyrazolo [1, 5-a] pyrimidine substituted diamide derivatives
A. K. Ajeesh Kumar, Yadav D. Bodke, Peter Serjious Lakra et al. · Medicinal Chemistry Research
|
22 Jan 2017 |
22 |
| 41 |
Synthesis Development of the Selective Estrogen Receptor Degrader (SERD) LSZ102 from a Suzuki Coupling to a C–H Activation Strategy
Markus Baenziger, Marcel Baierl, Krishnaswamy Devanathan et al. · Organic Process Research & Development
|
Jul 2020 |
21 |
| 42 |
Correlation of inducible nitric oxide synthase (iNOS) inhibition with TNF-α, caspase-1, FasL and TLR-3 in pathogenesis of rabies in mouse model
B. P. Madhu, Karam Pal Singh, M. Saminathan et al. · Virus Genes
|
21 Dec 2015 |
21 |
| 43 |
New azetidine-3-carbonyl-N-methyl-hydrazino derivatives of fluoroquinolones: synthesis and evaluation of antibacterial and anticancer properties
Gavara Govinda Rajulu, Halehatty S. Bhojya Naik, G. Charan Kumar et al. · Medicinal Chemistry Research
|
16 Nov 2013 |
21 |
| 44 |
Environmentally benign nucleophilic substitution reaction of arylalkyl halides in water using CTAB as the inverse phase transfer catalyst
Atul K. Godha, Jayaraman Thiruvengadam, Abhilash Viswanadhan et al. · New Journal of Chemistry
|
2019 |
20 |
| 45 |
Simultaneous exploration of TBAF·3H 2 O as a base as well as a solvating agent for the palladium catalyzed Suzuki cross-coupling of 4-methyl-7-nonafluorobutylsulfonyloxy coumarins under microwave irradiation
Muthipeedika Nibin Joy, Yadav D. Bodke, K.K. Abdul Khader et al. · Journal of Fluorine Chemistry
|
6 Jan 2016 |
20 |
| 46 |
Dehydration in water: solid-supported lipases as green catalysts for esterification
Rohan M. Thomas, Monica S. Lopez Lemus, Krithika Ganesh et al. · Green Chemistry
|
2024 |
19 |
| 47 |
E3 Ligases: a Potential Multi-Drug Target for Different Types of Cancers and Neurological Disorders
Konda Mani Saravanan, K. Muthu, Prabhakar Meera et al. · Future Medicinal Chemistry
|
19 Jan 2022 |
19 |
| 48 |
Copper-Catalyzed Asymmetric Reductions of Aryl/Heteroaryl Ketones under Mild Aqueous Micellar Conditions
David M. Fialho, Elham Etemadi‐Davan, Olivia C. Langner et al. · Organic Letters
|
27 Apr 2021 |
19 |
| 49 |
Sulfated polysaccharides from Caulerpa sertularioides: Extraction and evaluation of antioxidant, antibacterial, and immunological properties
Ravichandran Anjali, Subramanian Palanisamy, Manoharan Vinosha et al. · Industrial Crops and Products
|
29 Sep 2022 |
18 |
| 50 |
SARS-CoV-2 Mpro binding profile and drug-likeness of two novel thiazole derivatives: structural elucidation, DFT studies, ADME-T and molecular docking simulations
T.N. Lohith, Krishna Ravi Singh, Bienfait Kabuyaya Isamura et al. · Journal of Biomolecular Structure and Dynamics
|
28 Dec 2022 |
17 |