| 1 |
Role of LDH in tumor glycolysis: Regulation of LDHA by small molecules for cancer therapeutics
Dolly Sharma, Mamta Singh, Reshma Rani · Seminars in Cancer Biology
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9 Nov 2022 |
455 |
| 2 |
An Inhibitor of FtsZ with Potent and Selective Anti-Staphylococcal Activity
David J. Haydon, Neil R. Stokes, Rebecca Ure et al. · Science
Open access |
18 Sep 2008 |
453 |
| 3 |
Solid Dispersion as an Approach for Bioavailability Enhancement of Poorly Water-Soluble Drug Ritonavir
Shilpi Sinha, Mushir Ali, Sanjula Baboota et al. · AAPS PharmSciTech
Open access |
17 Mar 2010 |
234 |
| 4 |
Regio‐ and Chemoselective Reduction of Nitroarenes and Carbonyl Compounds over Recyclable Magnetic FerriteNickel Nanoparticles (Fe3O4Ni) by Using Glycerol as a Hydrogen Source
Manoj B. Gawande, Anuj Kumar Rathi, Paula S. Branco et al. · Chemistry - A European Journal
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30 Aug 2012 |
190 |
| 5 |
Targeting monocarboxylate transporters (MCTs) in cancer: How close are we to the clinics?
Mamta Singh, Julieta Afonso, Dolly Sharma et al. · Seminars in Cancer Biology
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24 Jan 2023 |
187 |
| 6 |
Magnetite-supported sulfonic acid: a retrievable nanocatalyst for the Ritter reaction and multicomponent reactions
Manoj B. Gawande, Anuj Kumar Rathi, Isabel Nogueira et al. · Green Chemistry
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2013 |
187 |
| 7 |
Irinotecan and its active metabolite, SN‐38: review of bioanalytical methods and recent update from clinical pharmacology perspectives
Ramesh Mullangi, Preeti Ahlawat, Nuggehally R. Srinivas · Biomedical Chromatography
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23 Oct 2009 |
181 |
| 8 |
Purple heart plant leaves extract-mediated silver nanoparticle synthesis: Optimization by Box-Behnken design
Md Saquib Hasnain, Md. Noushad Javed, Md Sabir Alam et al. · Materials Science and Engineering C
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15 Feb 2019 |
178 |
| 9 |
Medicinal importance, pharmacological activities, and analytical aspects of hispidulin: A concise report
Kanika Patel, Dinesh Kumar Patel · Journal of Traditional and Complementary Medicine
Open access |
10 Dec 2016 |
172 |
| 10 |
GSK3β: role in therapeutic landscape and development of modulators
Samiron Phukan, V. Venkatesh Babu, Akanksha Kannoji et al. · British Journal of Pharmacology
Open access |
20 Mar 2010 |
158 |
| 11 |
TGR5: an emerging bile acid G-protein-coupled receptor target for the potential treatment of metabolic disorders
Atul Kumar Tiwari, Pranab Maiti · Drug Discovery Today
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26 Feb 2009 |
120 |
| 12 |
Implication of Nano-Antioxidant Therapy for Treatment of Hepatocellular Carcinoma Using PLGA Nanoparticles of Rutin
Preeti Madhuri Pandey, Mahfoozur Rahman, Prakash Chandra Bhatt et al. · Nanomedicine
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22 Mar 2018 |
116 |
| 13 |
CREB is a critical regulator of normal hematopoiesis and leukemogenesis
Jerry C. Cheng, Kentaro Kinjo, Dejah R. Judelson et al. · Blood
Open access |
2 Nov 2007 |
115 |
| 14 |
Glioblastoma: Current Status, Emerging Targets, and Recent Advances
Amandeep Thakur, Chetna Faujdar, Ram Sharma et al. · Journal of Medicinal Chemistry
Open access |
5 Jul 2022 |
114 |
| 15 |
High yield synthesis of amine functionalized graphene oxide and its surface properties
Souvik Chakraborty, Saikat Saha, V.R. Dhanak et al. · RSC Advances
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2016 |
107 |
| 16 |
Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors
Victor S. Gehling et al. · ACS Medicinal Chemistry Letters
Open access |
16 Jul 2013 |
105 |
| 17 |
Creating an Antibacterial with in Vivo Efficacy: Synthesis and Characterization of Potent Inhibitors of the Bacterial Cell Division Protein FtsZ with Improved Pharmaceutical Properties
David J. Haydon, James M. Bennett, David Richard Brown et al. · Journal of Medicinal Chemistry
Open access |
28 Apr 2010 |
105 |
| 18 |
A small molecule inhibitor of Nicotinamide N-methyltransferase for the treatment of metabolic disorders
Aimo Kannt et al. · Scientific Reports
Open access |
20 Feb 2018 |
102 |
| 19 |
Oil based nanocarrier system for transdermal delivery of ropinirole: A mechanistic, pharmacokinetic and biochemical investigation
Adnan Azeem, Sushama Talegaonkar, Lalit Mohan Singh Negi et al. · International Journal of Pharmaceutics
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27 Oct 2011 |
98 |
| 20 |
An Improved Small-Molecule Inhibitor of FtsZ with Superior In Vitro Potency, Drug-Like Properties, and In Vivo Efficacy
Neil R. Stokes, Nicola Baker, James M. Bennett et al. · Antimicrobial Agents and Chemotherapy
Open access |
Nov 2012 |
98 |
| 21 |
Sustainable Utility of Magnetically Recyclable Nano-Catalysts in Water: Applications in Organic Synthesis
Manoj B. Gawande, Anuj Kumar Rathi, Paula S. Branco et al. · Applied Sciences
Open access |
25 Oct 2013 |
96 |
| 22 |
First application of core-shell Ag@Ni magnetic nanocatalyst for transfer hydrogenation reactions of aromatic nitro and carbonyl compounds
Manoj B. Gawande, Huizhang Guo, Anuj Kumar Rathi et al. · RSC Advances
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15 Nov 2012 |
93 |
| 23 |
PAD4: pathophysiology, current therapeutics and future perspective in rheumatoid arthritis
Sindhu Koushik, Nivedita Joshi, Shruthi Nagaraju et al. · Expert Opinion on Therapeutic Targets
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16 Feb 2017 |
86 |
| 24 |
Could MM-GBSA be accurate enough for calculation of absolute protein/ligand binding free energies?
Chandrika Mulakala, Vellarkad N. Viswanadhan · Journal of Molecular Graphics and Modelling
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18 Sep 2013 |
86 |
| 25 |
A Recyclable Ferrite–Co Magnetic Nanocatalyst for the Oxidation of Alcohols to Carbonyl Compounds
Manoj B. Gawande, Anuj Kumar Rathi, Isabel Nogueira et al. · ChemPlusChem
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10 Aug 2012 |
84 |
| 26 |
GLUT and HK: Two primary and essential key players in tumor glycolysis
Dhiraj Yadav, Anubha Yadav, Sujata Bhattacharya et al. · Seminars in Cancer Biology
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15 Mar 2024 |
82 |
| 27 |
New insights into the medicinal importance, physiological functions and bioanalytical aspects of an important bioactive compound of foods ‘Hyperin’: Health benefits of the past, the present, the future
Kanika Patel, Vikas Kumar, Mahfoozur Rahman et al. · Beni-Suef University Journal of Basic and Applied Sciences
Open access |
Jun 2017 |
82 |
| 28 |
Design, synthesis and structure–activity relationships of substituted oxazole–benzamide antibacterial inhibitors of FtsZ
Neil R. Stokes et al. · Bioorganic & Medicinal Chemistry Letters
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13 Nov 2013 |
80 |
| 29 |
Synthesis, anti-tubercular activity and 3D-QSAR study of coumarin-4-acetic acid benzylidene hydrazides
Atul T. Manvar, Alpeshkumar K. Malde, Jitender Kumar Verma et al. · European Journal of Medicinal Chemistry
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31 Jan 2008 |
79 |
| 30 |
PLK4: a link between centriole biogenesis and cancer
Radhika Radha Maniswami, Seema Prashanth, Archana Venkataramana Karanth et al. · Expert Opinion on Therapeutic Targets
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24 Nov 2017 |
75 |
| 31 |
Emerging role of SETDB1 as a therapeutic target
Archana Venkataramana Karanth, Radhika Radha Maniswami, Seema Prashanth et al. · Expert Opinion on Therapeutic Targets
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11 Jan 2017 |
72 |
| 32 |
Alleviation of arthritis through prevention of neutrophil extracellular traps by an orally available inhibitor of protein arginine deiminase 4
Chandru Gajendran, Shoichi Fukui, Naveen M. Sadhu et al. · Scientific Reports
Open access |
23 Feb 2023 |
69 |
| 33 |
A comprehensive study on regulatory requirements for development and filing of generic drugs globally
Shweta Handoo, Deepak Khera, PrafullaKumar Nandi et al. · International Journal of Pharmaceutical Investigation
Open access |
2012 |
69 |
| 34 |
SIGNAL TRANSDUCTION PATHWAYS LINKING THE ACTIVATION OF ALVEOLAR MACROPHAGES WITH THE RECRUITMENT OF NEUTROPHILS TO LUNGS IN CHRONIC OBSTRUCTIVE PULMONARY DISEASE
Vidyasaral Murugan, Michael J. Peck · Experimental Lung Research
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2009 |
68 |
| 35 |
MPX-004 and MPX-007: New Pharmacological Tools to Study the Physiology of NMDA Receptors Containing the GluN2A Subunit
Robert A. Volkmann, Christopher M. Fanger, David R. Anderson et al. · PLoS ONE
Open access |
Feb 2016 |
65 |
| 36 |
The Discovery, Preclinical, and Early Clinical Development of Potent and Selective GPR40 Agonists for the Treatment of Type 2 Diabetes Mellitus (LY2881835, LY2922083, and LY2922470)
Chafiq Hamdouchi et al. · Journal of Medicinal Chemistry
Open access |
17 Oct 2016 |
62 |
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Insights into the Targeting Potential of Thymoquinone for Therapeutic Intervention Against Triple-negative Breast Cancer
Md. Abul Barkat, Harshita, Javed Ahmad et al. · Current Drug Targets
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5 Jan 2018 |
60 |
| 38 |
Simultaneous determination of atorvastatin, amlodipine, ramipril and benazepril in human plasma by LC‐MS/MS and its application to a human pharmacokinetic study
Nageswara Rao Pilli, Jaswanth Kumar Inamadugu, Ramesh Mullangi et al. · Biomedical Chromatography
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13 Jul 2010 |
60 |
| 39 |
Soluble starch-blended Ca 2+ -Zn 2+ -alginate composites-based microparticles of aceclofenac: Formulation development and in vitro characterization
Amit Kumar Nayak, Jadupati Malakar, Dilipkumar Pal et al. · Future Journal of Pharmaceutical Sciences
Open access |
18 Mar 2018 |
59 |
| 40 |
Identification of Allosteric PIF‐Pocket Ligands for PDK1 using NMR‐Based Fragment Screening and 1H‐15N TROSY Experiments
Brian J. Stockman, Michael Kothe, Darcy Kohls et al. · Chemical Biology & Drug Design
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22 Jan 2009 |
58 |
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Emergence in the functionalized carbon nanotubes as smart nanocarriers for drug delivery applications
Sarwar Beg, Mahfoozur Rahman, Atul Jain et al. · Elsevier eBooks
Book chapterOpen access |
2018 |
57 |
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Synthesis and Evaluation of the 2-Aminothiazoles as Anti-Tubercular Agents
Edward A. Kesicki, Mai Ann Bailey, Yulia Ovechkina et al. · PLoS ONE
Open access |
12 May 2016 |
57 |
| 43 |
Nanosuspension-Based Aloe vera Gel of Silver Sulfadiazine with Improved Wound Healing Activity
Md. Abul Barkat, Harshita, Iqbal Ahmad et al. · AAPS PharmSciTech
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5 Jun 2017 |
56 |
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The synthesis and evaluation of triazolopyrimidines as anti-tubercular agents
Edison S. Zuniga, Aaron Korkegian, Steven F. Mullen et al. · Bioorganic & Medicinal Chemistry
Open access |
19 May 2017 |
56 |
| 45 |
Quantitation of VEGFR2 (vascular endothelial growth factor receptor) inhibitors – review of assay methodologies and perspectives
Kuldeep Kumar Sharma, P. S. Suresh, Ramesh Mullangi et al. · Biomedical Chromatography
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26 Nov 2014 |
56 |
| 46 |
A classification model for blood brain barrier penetration
Manvi Singh, Reshmi Divakaran, Leela Sarath Kumar Konda et al. · Journal of Molecular Graphics and Modelling
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20 Dec 2019 |
55 |
| 47 |
High-Affinity Alkynyl Bisubstrate Inhibitors of Nicotinamide N -Methyltransferase (NNMT)
Rocco L. Policarpo, Ludovic Decultot, Elizabeth May et al. · Journal of Medicinal Chemistry
Open access |
7 Oct 2019 |
55 |
| 48 |
Silica gel promoted environment-friendly synthesis of 2,3-disubstituted 4-thiazolidinones
Manoj P. Thakare, Puneet Kumar, Naresh Kumar et al. · Tetrahedron Letters
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11 Mar 2014 |
54 |
| 49 |
Development and validation of a highly sensitive and robust LC‐ESI‐MS/MS method for simultaneous quantitation of simvastatin acid, amlodipine and valsartan in human plasma: application to a clinical pharmacokinetic study
Addepalli Venkata Ramani, Pinaki Sengupta, Ramesh Mullangi · Biomedical Chromatography
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10 Mar 2009 |
54 |
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Pose Prediction Accuracy in Docking Studies and Enrichment of Actives in the Active Site of GSK-3β
Pravin Kumar Gadakar, Samiron Phukan, and Prasanna Dattatreya et al. · Journal of Chemical Information and Modeling
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20 Jun 2007 |
53 |