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Most cited papers in Asymmetric Synthesis and Catalysis

Asymmetric Synthesis and Catalysis

What are the most cited papers in Asymmetric Synthesis and Catalysis?

The most cited paper in Asymmetric Synthesis and Catalysis is "Aryl−Aryl Bond Formation One Century after the Discovery of the Ullmann Reaction" (Jwanro Hassan, Marc Sévignon, Christel Gozzi et al., 2002), with 3,659 citations. Next come "Asymmetric Transition Metal-Catalyzed Allylic Alkylations" (3,206) and "Natural Products as Sources of New Drugs over the Period 1981−2002" (3,095).

Showing 50 of 100 papers. Every paper with more than 1,012 citations is listed.

Most cited papers, sortable by citations and release date
#Paper
1 Aryl−Aryl Bond Formation One Century after the Discovery of the Ullmann Reaction Jwanro Hassan, Marc Sévignon, Christel Gozzi et al. · Chemical Reviews Review 8 Mar 2002 3,659
2 Asymmetric Transition Metal-Catalyzed Allylic Alkylations Barry M. Trost, David L. Van Vranken · Chemical Reviews Review 1996 3,206
3 Natural Products as Sources of New Drugs over the Period 1981−2002 David J. Newman, Gordon M. L. Cragg, Kenneth M. Snader · Journal of Natural Products 12 Jun 2003 3,095
4 CH Bond Functionalization: Emerging Synthetic Tools for Natural Products and Pharmaceuticals Junichiro Yamaguchi, Atsushi D. Yamaguchi, Kenichiro Itami · Angewandte Chemie International Edition 6 Aug 2012 2,994
5 Proline-Catalyzed Direct Asymmetric Aldol Reactions Benjamin List, Richard Alan Lerner, Carlos F. Barbas · Journal of the American Chemical Society 26 Feb 2000 2,868
6 Asymmetric Transition-Metal-Catalyzed Allylic Alkylations: Applications in Total Synthesis Barry M. Trost, Matthew L. Crawley · Chemical Reviews Review 21 Jun 2003 2,854
7 Asymmetric Enamine Catalysis Santanu Mukherjee, Jung Woon Yang, S.D. Hoffmann et al. · Chemical Reviews Review Dec 2007 2,854
8 Palladium‐Catalyzed Cross‐Coupling Reactions in Total Synthesis Kyriacos Costa Nicolaou, Paul G. Bulger, David Šarlah · Angewandte Chemie International Edition 30 Jun 2005 2,714
9 Atom Economy—A Challenge for Organic Synthesis: Homogeneous Catalysis Leads the Way Barry M. Trost · Angewandte Chemie International Edition in English 21 Feb 1995 2,602
10 In the Golden Age of Organocatalysis Peter I. Dalko, Lionel Moisan · Angewandte Chemie International Edition 29 Sep 2004 2,586
11 New Chiral Phosphorus Ligands for Enantioselective Hydrogenation Wenjun Tang, Xumu Zhang · Chemical Reviews Review 6 Jun 2003 2,567
12 The advent and development of organocatalysis David W. C. MacMillan · Nature Sep 2008 2,407
13 Reagents for Organic Synthesis Richard C. Larock · Journal of Organometallic Chemistry May 1976 2,346
14 Stronger Brønsted Acids Takahiko Akiyama · Chemical Reviews Review 6 Nov 2007 2,311
15 Organic Reactions in Aqueous Media with a Focus on Carbon−Carbon Bond Formations: A Decade Update Chao‐Jun Li · Chemical Reviews Review 23 Jul 2005 2,245
16 Effect of Chlorpromazine or Haloperidol on Formation of 3‐Methoxytyramine and Normetanephrine in Mouse Brain Arvid Carlsson, Margit Lindqvist · Acta Pharmacologica et Toxicologica Sep 1963 2,157
17 Iron-Catalyzed Reactions in Organic Synthesis Carsten Bolm, Julien Legros, Jacques Le Paih et al. · Chemical Reviews Review 19 Nov 2004 2,144
18 Practical Methodologies for the Synthesis of Indoles Guy R. Humphrey, Jeffrey T. Kuethe · Chemical Reviews Review 7 Jun 2006 2,142
19 Complete Field Guide to Asymmetric BINOL-Phosphate Derived Brønsted Acid and Metal Catalysis: History and Classification by Mode of Activation; Brønsted Acidity, Hydrogen Bonding, Ion Pairing, and Metal Phosphates Dixit Parmar, Erli Sugiono, Sadiya Raja et al. · Chemical Reviews ReviewOpen access 9 Sep 2014 2,107
20 Recent advances in olefin metathesis and its application in organic synthesis Robert Howard Grubbs, Sukbok Chang · Tetrahedron Apr 1998 2,101
21 Cascade Reactions in Total Synthesis Kyriacos Costa Nicolaou, David J. Edmonds, Paul G. Bulger · Angewandte Chemie International Edition 30 Oct 2006 2,093
22 Asymmetric Catalysis: Science and Opportunities (Nobel Lecture) Copyright© The Nobel Foundation 2002. We thank the Nobel Foundation, Stockholm, for permission to print this lecture. Ryōji Noyori · Angewandte Chemie International Edition 17 Jun 2002 2,042
23 Frustrated Lewis Pairs: Metal‐free Hydrogen Activation and More Douglas W. Stephan, Gerhard Erker · Angewandte Chemie International Edition 18 Dec 2009 1,996
24 Asymmetric 1,3-Dipolar Cycloaddition Reactions Kurt V. Gothelf, Karl Anker Jørgensen · Chemical Reviews Review 14 Mar 1998 1,913
25 Asymmetric Catalysis by Chiral Hydrogen‐Bond Donors Mark S. Taylor, Eric N. Jacobsen · Angewandte Chemie International Edition 21 Feb 2006 1,908
26 Stereoselective Cyclopropanation Reactions H. Lebel, Jean-François Marcoux, Carmela Molinaro et al. · Chemical Reviews Review Apr 2003 1,796
27 A Medicinal Chemist’s Guide to Molecular Interactions Caterina Bissantz, Bernd Kuhn, Martin Ståhl · Journal of Medicinal Chemistry Open access 26 Mar 2010 1,760
28 New Strategies for Organic Catalysis: The First Highly Enantioselective Organocatalytic Diels−Alder Reaction Kateri A. Ahrendt, Christopher J. Borths, David W. C. MacMillan · Journal of the American Chemical Society 15 Apr 2000 1,690
29 Enantioselective Mannich‐Type Reaction Catalyzed by a Chiral Brønsted Acid Takahiko Akiyama, Junji Itoh, Koji Yokota et al. · Angewandte Chemie International Edition 9 Mar 2004 1,670
30 Stereoselective Organic Reactions in Water Ulf M. Lindström · Chemical Reviews Review 19 Jun 2002 1,643
31 1,2-Amino Alcohols and Their Heterocyclic Derivatives as Chiral Auxiliaries in Asymmetric Synthesis David J. Ager, Indra Prakash, David R. Schaad · Chemical Reviews Review 1996 1,627
32 Asymmetric Organocatalytic Domino Reactions Dieter Enders, Christoph Grondal, Matthias R. M. Hüttl · Angewandte Chemie International Edition 16 Jan 2007 1,622
33 Chiral Brønsted Acid-Catalyzed Direct Mannich Reactions via Electrophilic Activation Daisuke Uraguchi, Masahiro Terada · Journal of the American Chemical Society 9 Apr 2004 1,611
34 Modern Organic Synthesis with α-Diazocarbonyl Compounds Alan Ford, Hugues Miel, Aoife Ring et al. · Chemical Reviews Review 18 Aug 2015 1,607
35 Isatins As Privileged Molecules in Design and Synthesis of Spiro-Fused Cyclic Frameworks Girija Shankar Singh, Zelalem Yibralign Desta · Chemical Reviews Review 6 Sep 2012 1,595
36 Donor−Acceptor-Substituted Cyclopropane Derivatives and Their Application in Organic Synthesis Hans‐Ulrich Reißig, Reinhold Zimmer · Chemical Reviews Review 21 Feb 2003 1,592
37 Organocatalytic cascade reactions as a new tool in total synthesis Christoph Grondal, Matthieu Jeanty, Dieter Enders · Nature Chemistry 19 Feb 2010 1,583
38 Catalytic Enantioselective Addition to Imines Shū Kobayashi, Haruro Ishitani · Chemical Reviews Review 20 Apr 1999 1,570
39 C−F Bond Activation in Organic Synthesis Hideki Amii, Kenji Uneyama · Chemical Reviews Review 30 Mar 2009 1,547
40 Metal‐Catalyzed Enantioselective Allylation in Asymmetric Synthesis Zhan Ling Lu, Shengming Ma · Angewandte Chemie International Edition 29 Oct 2007 1,507
41 The osmium-catalyzed asymmetric dihydroxylation: a new ligand class and a process improvement Karl Barry Sharpless, Willi M. Amberg, Youssef L. Bennani et al. · The Journal of Organic Chemistry May 1992 1,483
42 Some Typical Advances in the Synthetic Applications of Allenes Shengming Ma · Chemical Reviews Review 9 Jun 2005 1,482
43 Privileged Chiral Catalysts Tehshik P. Yoon, Eric N. Jacobsen · Science 13 Mar 2003 1,465
44 Construction of Spiro[pyrrolidine‐3,3′‐oxindoles] − Recent Applications to the Synthesis of Oxindole Alkaloids Christiane Marti, Erick M. Carreira · European Journal of Organic Chemistry Jun 2003 1,454
45 Rhodium-Catalyzed Asymmetric 1,4-Addition and Its Related Asymmetric Reactions Tamio Hayashi, Kaori Yamasaki · Chemical Reviews Review 24 Jul 2003 1,437
46 Iminium Catalysis Anniina Erkkilä, Inkeri Majander, Petri M. Pihko · Chemical Reviews Review Dec 2007 1,435
47 Enantioselective Michael Reaction of Malonates to Nitroolefins Catalyzed by Bifunctional Organocatalysts Tomotaka Okino, Yasutaka Hoashi, Yoshiji Takemoto · Journal of the American Chemical Society 30 Sep 2003 1,422
48 Enamine-Based Organocatalysis with Proline and Diamines: The Development of Direct Catalytic Asymmetric Aldol, Mannich, Michael, and Diels−Alder Reactions Wolfgang Notz, Fujie Tanaka, Carlos F. Barbas · Accounts of Chemical Research 10 Jul 2004 1,369
49 Asymmetric Catalysis with Water: Efficient Kinetic Resolution of Terminal Epoxides by Means of Catalytic Hydrolysis Makoto Tokunaga, Jay F. Larrow, Fumitoshi Kakiuchi et al. · Science 15 Aug 1997 1,365
50 Dearomatization Strategies in the Synthesis of Complex Natural Products Stephane Philippe Roche, John A. Jr. Porco · Angewandte Chemie International Edition Open access 19 Apr 2011 1,354

Citations are OpenAlex's own counts, from its 2026-09-23 snapshot, so the ranking can differ from Google Scholar or Web of Science. A paper is listed for a field when OpenAlex files it under one of the field's topics; retracted papers and papers whose citation count cannot be traced to citing works are left out, and a preprint and the article it became are shown once. Release dates are OpenAlex's: where a source gave only a month or a year, that is what is shown. How the lists are chosen.